Albendazole yog ib qho tshuaj anthelmintic hluavtaws uas yog ib feem ntawm pawg benzimidazole-derivatives nrog kev ua haujlwm tawm tsam ntau hom kab thiab ntawm qib siab dua kuj tawm tsam cov neeg laus ntawm cov kab mob siab.
Albendazole ua ke nrog eelworm lub microtubule protein thiab ua lub luag haujlwm. Tom qab albenzene ua ke nrog β-tubulin, nws tuaj yeem tiv thaiv dimerization ntawm albenzene thiab α tubulin sib sau ua ke rau hauv microtubules. Microtubules yog cov qauv yooj yim ntawm ntau lub cell units. Albendazole qhov sib raug zoo rau nematodes tubulin yog siab dua qhov sib raug zoo ntawm mammalian tubulin, yog li kev lom rau mammalian yog me me.
Kev tiv thaiv thiab kho cov kab mob worm hauv cov nyuj thiab nyuj xws li:
Cov kab mob gastrointestinal:Bunostomum, Cooperia, Chabertia, Haemonchus, Nematodirus, Oesophagostomum, Ostertagia, Strongyloides thiab Trichostrongylus spp.
Cov kab mob ntsws:Dictyocaulus viviparus thiab D. filaria.
Kab mob Tapeworms:Monieza spp.
Kab mob siab:cov neeg laus Fasciola hepatica.
Albendazole kuj tseem muaj cov nyhuv tua oviduct.
Kev tswj hwm hauv 45 hnub thawj zaug ntawm kev cev xeeb tub.
Cov tshuaj tiv thaiv hypersensitivity.
Rau kev tswj hwm qhov ncauj.
Rau cov kab mob roundworms, tapeworms:
Nyuj / twm / nees / yaj / tshis: 5mg / kg lub cev hnyav
Aub / miv: 10 txog 25mg / kg lub cev hnyav
Rau cov flukes:
Nyuj/twm: 10mg/kg lub cev hnyav
Yaj/tshis: 7.5mg/kg lub cev hnyav
Cov menyuam nyuj thiab nyuj: 1 bolus rau txhua 300 kg ntawm qhov hnyav.
Rau cov kab mob siab:
1 bolus rau txhua 250 kg ntawm qhov hnyav.
Khaws cia kom deb ntawm cov menyuam yaus.
3 xyoos.
- Rau nqaij:12 hnub.
- Rau cov mis nyuj:4 hnub.
Khaws cia rau qhov chaw txias thiab qhuav uas tiv thaiv kom tsis txhob muaj teeb.